ANTHACAINE contains Lignocaine (Lidocaine) which belongs to a group of medicines called local anaesthetics which produces a temporary loss of feeling or numbness of the area. It is used before certain types of examination, production of anesthesia of accessible mucous membranes of the oropharynx and for the temporary relief of pain associated with minor burns, sunburn, abrasions of the skin, insect bites and hemorrhoids.
Lignocaine (Lidocaine) is a potent local anaesthetic of the amide type. Like other local anaesthetics, it prevents both the generation and conduction of nerve impulses by slowing depolarisation. This results from blocking of the large transient increase in permeability of the cell membrane to sodium ions that follows initial depolarisation of the membrane. It acts reversible blockade of impulse propagation by prevention of sodium flux. As a local anesthetic, lidocaine blocks initiation and conduction of nerve impulses by decreasing the permeability of the nerve cell membrane to sodium ions.
Before using ANTHACAINE tell your doctor if you have liver, kidney or heart problems, are pregnant or breastfeeding. Your doctor will give the correct dose depends on your child’s age and body weight. The common side effects are dizziness, irritation, redness at the application site. Avoid contact with eyes.
Used to,
ANTHACAINE blocks nerve transmission, when applied to a limited area of the body, which they bind to the sodium channels in the nerve membrane and prevent the entry of sodium ions in response to the membrane’s depolarization.
Always use ANTHACAINE as prescribed by your doctor. Your doctor will give dose depends on type of pain. Check the label for direction before use.
Dizziness:
Get up and move around to feel awake, take small naps to edge off the sleepiness. Give your eyes a break to avoid fatigue and eat a healthy food to boost energy.
ANTHACAINE should be used with caution in pregnant women. Discuss the risks and benefits with your doctor.
ANTHACAINE should be used with caution during breastfeeding. Discuss the risks and benefits with your doctor.
ANTHACAINE may affect your ability to drive or handle any machines depending on where and how it is used.
ANTHACAINE should be used with caution in patients suffering from active kidney diseases. Consult your doctor for advice.
ANTHACAINE should be used with caution in patients suffering from active liver diseases. Consult your doctor for advice.
Tell your doctor if you are allergic (hypersensitive) to Lignocaine (Lidocaine).
ANTHACAINE is not recommended in patients with severe slow heartbeat or any other active heart diseases. Consult your doctor for advice.
Inform your doctor if you have or had,
Inform your doctor if you are using or have recently taken any other medicines, including medicines obtained without a prescription or the following,
Drug | : | Lignocaine (Lidocaine) |
Pharmacological Category | : | Antiarrhythmic agent |
Therapeutic Indication | : | Topical anesthesia of the mucous membranes of the respiratory tract and painful oral conditions |
Dosage Forms | : | Injection (Solution, Intraspinal, Intravenous), Cream, Solution, Spray |
Store below 20-25°C and keep out of reach of children.
When does ANTHACAINE starts to work?
It starts working within 5 minutes after you apply it, the pain relief effect lasts about 4 hours for wounds caused by burning.
Does ANTHACAINE use during pregnancy?
It should be used with caution during pregnancy, or if you are trying to get pregnant. Consult your doctor for advice.
Does ANTHACAINE cause dizziness?
It may cause drowsiness or dizziness, do not drive or handle any machines if you experience these reactions.
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